Amauromine |
رقم الكتالوجGC42778 |
Amauromine is a neutral antagonist of the cannabinoid (CB) receptor CB1 that is selective for CB1 (Ki = 178 nM; Kb = 66.6 nM) over CB2, with no activity at CB2 receptors at concentrations up to 10 μM.
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Cas No.: 88360-87-6
Sample solution is provided at 25 µL, 10mM.
Amauromine is a neutral antagonist of the cannabinoid (CB) receptor CB1 that is selective for CB1 (Ki = 178 nM; Kb = 66.6 nM) over CB2, with no activity at CB2 receptors at concentrations up to 10 µM. It is also an antagonist of GPR18 (IC50 = 3.74 µM). Amauromine has vasodilatory activity.
Average Rating: 5
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