NaV1.7 inhibitor-1 |
| رقم الكتالوجGC36698 |
مثبط NaV1.7 - 1 هو مثبط فعال لقناة الصوديوم ذات الجهد الكهربائي (NaV) 1.7 مع IC بمقدار 0.6 نانومتر لـ hNaV1.7 ، ويظهر انتقائية 80 ضعفًا مقابل hNaV1.5
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Cas No.: 1494585-79-3
Sample solution is provided at 25 µL, 10mM.
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NaV1.7 inhibitor-1 is an efficacious voltage-gated sodium channel (NaV) 1.7 inhibitor with an IC50 of 0.6 nM for hNaV1.7, exhibits 80-fold selectivity versus hNaV1.5[1]. IC50: 0.6 nM (hNaV1.7)[1]
[1]. Sun S, Identification of Selective Acyl Sulfonamide-Cycloalkylether Inhibitors of the Voltage-GatedSodium Channel (NaV) 1.7 with Potent Analgesic Activity. J Med Chem. 2019 Jan 24;62(2):908-927.
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