GX 201 |
| رقم الكتالوجGC50707 |
GX 201 هو مثبط انتقائي NaV1.7 ، مع IC 50 \u003c3.2 نانومتر لـ hNaV1.7.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1788071-27-1
Sample solution is provided at 25 µL, 10mM.
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Potent and selective Nav1.7 blocker (IC50 = 3.2 nM). Exhibits 10x selectivity for Nav1.7 over Nav1.1, Nav1.2, and Nav1.6 channels. Displays prolonged residency time on the Nav1.7 channel. Chronic dosing increases compound potency ~10-fold and provides efficacy that persists after the compound has cleared from plasma. Suppresses neuropathic pain in a mouse diabetic neuropathy model. Analgesic.
Average Rating: 5 (Based on Reviews and 7 reference(s) in Google Scholar.)
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