mAChR antagonist 1 |
| رقم الكتالوجGC71334 |
mAChR antagonist 1 (مركب 4a) هو مضاد mAChR مع قيم Ki من 255 نانومتر و 121 نانومتر و 158 نانومتر و 255 نانومتر للأنواع الفرعية M1 و M3 و M4 و M5 على التوالي.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 101491-79-6
Sample solution is provided at 25 µL, 10mM.
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mAChR antagonist 1 (compound 4a) is a mAChR antagonist with Ki values of 255 nM, 121 nM, 158 nM, and 255 nM for M1, M3, M4, and M5 subtype, respectively.
References:
[1]. Marlon Millard, et al. Design, synthesis and preclinical evaluation of muscarine receptor antagonists via a scaffold-hopping approach. Eur J Med Chem. 2023 Oct 21:262:115891.
Review for mAChR antagonist 1
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Review for mAChR antagonist 1
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