SER-601 |
| رقم الكتالوجGC18867 |
A selective CB2 receptor agonist
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1048038-90-9
Sample solution is provided at 25 µL, 10mM.
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SER-601 is a potent and selective peripheral cannabinoid (CB2) receptor agonist with 190-fold selectivity for CB2 over the central CB1 receptor (Kis = 6.3 and 1,220 nM, respectively). At 3 mg/kg, SER-601 has analgesic effects in a formalin-induced nocifensive study in mice without cannabis-like behavioral effects due to its low affinity for the CB1 receptor. SER-601 also has antidiabetic effects. Two to four week exposure to SER-601 ameliorates insulin resistance in vivo and increases insulin secretion and accumulation in pancreatic islets isolated from high-fat diet/streptozotocin (HFD/STZ)-induced diabetic mice.
Review for SER-601
Average Rating: 5 (Based on Reviews and 19 reference(s) in Google Scholar.)
Review for SER-601
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