SYM 2081 |
رقم الكتالوجGC16101 |
SYM 2081 عبارة عن مركب ترابطي عالي التقارب وناشط انتقائي قوي لمستقبلات كاينات ، ويثبط [3H] - الارتباط الحركي مع IC50 من 35 نانومتر ، انتقائية تقريبًا 3000 و 200 ضعف لمستقبلات كاينات على مستقبلات AMPA و NMDA على التوالي [1 ]
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Cas No.: 31137-74-3
Sample solution is provided at 25 µL, 10mM.
SYM 2081 is a high-affinity ligand and potent, selective agonist of kainate receptors, inhibits [3H]-kainate binding with an IC50 of 35 nM, almost 3000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively[1].
References:
[1]. Lee JY, et al. Furthering pharmacological and physiological assessment of the glutamatergic receptors at the Drosophila neuromuscular junction. Comp Biochem Physiol C Toxicol Pharmacol. 2009 Nov;150(4):546-57.
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