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CB1R Allosteric modulator 3

Catalog No.GC71115

CB1R Allosteric modulator 3 is a CB1R positive allosteric modulator.

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CB1R Allosteric modulator 3 Chemical Structure

Cas No.: 2633686-36-7

Size Price Stock Qty
5 mg
$90.00
In stock
10 mg
$153.00
In stock

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents
CB1R Allosteric modulator 3 is a CB1R positive allosteric modulator. CB1R Allosteric modulator 3 has potent inhibition of cAMP and β-Arrestin with EC50 values of 0.018 μM and 1.241 μM, respectively.

CB1R Allosteric modulator 3 (compound 44) (0.10 nM-10 μM, 30 min) has potent inhibition of cAMP and β-Arrestin with EC50 values of 0.018 μM and 1.241 μM, respectively[1].
CB1R Allosteric modulator 3 can enhance CB1R ago-PAM activity because of small lipophilic functional groups on the ortho-position of the GAT211 site-III phenyl ring[1].

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