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Dasatinib analog-1

Catalog No.GC71411

Dasatinib analog-1 (compound 5826) inhibits CYP3A4 viability with a Ki value of 5.4 μM.

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Dasatinib analog-1 Chemical Structure

Cas No.: 1174416-41-1

Size Price Stock Qty
5 mg
$171.00
In stock
10 mg
$279.00
In stock
25 mg
$563.00
In stock

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents
Dasatinib analog-1 (compound 5826) inhibits CYP3A4 viability with a Ki value of 5.4 μM. Dasatinib analog-1 blocks the formation of glutathione adducts.

References:
[1]. Xiaohai Li, et al. Characterization of dasatinib and its structural analogs as CYP3A4 mechanism-based inactivators and the proposed bioactivation pathways. Drug Metab Dispos. 2009, 37, 6.

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