AM 12 |
Katalog-Nr.GC50475 |
TRPC5 inhibitor
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2387510-84-9
Sample solution is provided at 25 µL, 10mM.
TRPC5 inhibitor (IC50 = 0.28 μM); Galangin derivative. Exhibits some selectivity for TRPC5 over TRPC2, 3 and 4. Inhibits effects of TRPC5 activator (-)-Englerin A, but potentiates effects of physiological activators Sphingosine-1-phosphate and LPC.
Naylor et al (2016) Natural and synthetic flavonoid modulation of TRPC5 channels. Br.J.Pharmacol. 173 562 PMID:26565375
Average Rating: 5
(Based on Reviews and 21 reference(s) in Google Scholar.)GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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