mAChR antagonist 1 |
| Katalog-Nr.GC71334 |
mAChR antagonist 1 (Verbindung 4a) ist ein mAChR-Antagonist mit Ki-Werten von 255 nM, 121 nM, 158 nM und 255 nM für M1, M3, M4 und M5 Subtypen.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 101491-79-6
Sample solution is provided at 25 µL, 10mM.
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mAChR antagonist 1 (compound 4a) is a mAChR antagonist with Ki values of 255 nM, 121 nM, 158 nM, and 255 nM for M1, M3, M4, and M5 subtype, respectively.
References:
[1]. Marlon Millard, et al. Design, synthesis and preclinical evaluation of muscarine receptor antagonists via a scaffold-hopping approach. Eur J Med Chem. 2023 Oct 21:262:115891.
Review for mAChR antagonist 1
Average Rating: 5 (Based on Reviews and 30 reference(s) in Google Scholar.)
Review for mAChR antagonist 1
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