rel-VU6021625 |
| Katalog-Nr.GC71468 |
rel-VU6021625 ist die weniger aktive relative Konfiguration von VU6021625.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2307718-96-1
Sample solution is provided at 25 µL, 10mM.
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rel-VU6021625 is the less active relative configuration of VU6021625 . VU6021625 is a potent and selective mAChR M4 antagonist with IC50 values of 0.44 nM and 57 nM for human M4, rat M4, respectively.
References:
[1]. Moehle MS, et al. Discovery of the First Selective M4 Muscarinic Acetylcholine Receptor Antagonists with in Vivo Antiparkinsonian and Antidystonic Efficacy. ACS Pharmacol Transl Sci. 2021 Aug 2;4(4):1306-1321.
Review for rel-VU6021625
Average Rating: 5 (Based on Reviews and 30 reference(s) in Google Scholar.)
Review for rel-VU6021625
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