Cyproheptadine (hydrochloride hydrate) |
Katalog-Nr.GC43353 |
Cyproheptadin (Hydrochloridhydrat) ist ein Antihistaminikum und ein Antagonist von Serotonin und Histamin2.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 41354-29-4
Sample solution is provided at 25 µL, 10mM.
Cyproheptadine is a first-generation antihistamine that potently antagonizes the histamine H1 receptor (pKi = 9.42). It also antagonizes serotonin and muscarinic receptors at nanomolar concentrations. Cyproheptadine also inhibits the lysine methyltransferase SET7/9 (IC50 = 1 µM), suppressing the expression of estrogen receptor α in human breast cancer MCF-7 cells.
Average Rating: 5
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