(R)-ZINC 3573 |
Katalog-Nr.GC50426 |
MRGPRX2 agonist
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2089389-15-9
Sample solution is provided at 25 µL, 10mM.
Mas-related G protein-coupled receptor X2 (MRGPRX2) agonist (EC50 = 0.74 μM). Displays selectivity for MRGPRX2 over 350 other GPCRs, including MRGPRX1. Induces intracellular calcium release and degranulation in LAD2 mast cells in vitro. Negative control (S)-ZINC 3573 also available.
Lansu et al (2017) In silico design of novel probes for the atypical opioid receptor MRGPRX2. Nat.Chem.Biol. 13 529 PMID:28288109
Average Rating: 5
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