RXR antagonist 1 |
| Katalog-Nr.GC70895 |
RXR antagonist 1 (Verbindung 6a) ist ein Retinoid-X-Rezeptor (RXR)-Modulator.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 3010910-40-1
Sample solution is provided at 25 µL, 10mM.
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RXR antagonist 1 (compound 6a) shows potent RXR-antagonistic activities at 1 μM[1].
RXR antagonist 1 shows competitive binding to the LBP in hRXRα-LBD, with Ki of 0.384 ± 0.072, Kd of 0.277 ± 0.038, and Ki/Kd of 1.39[1].
The cell permeability of RXR antagonist 1 shows no correlation with RXR-antagonistic activity[1].
Average Rating: 5 (Based on Reviews and 30 reference(s) in Google Scholar.)
GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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