SYM 2081 |
| Katalog-Nr.GC16101 |
SYM 2081 ist ein hochaffiner Ligand und potenter, selektiver Agonist von Kainatrezeptoren, hemmt die [3H]-Kainatbindung mit einer IC50 von 35 nM, fast 3000- und 200-facher SelektivitÄt fÜr Kainatrezeptoren gegenÜber AMPA- bzw. NMDA-Rezeptoren[1 ].
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 31137-74-3
Sample solution is provided at 25 µL, 10mM.
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SYM 2081 is a high-affinity ligand and potent, selective agonist of kainate receptors, inhibits [3H]-kainate binding with an IC50 of 35 nM, almost 3000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively[1].
References:
[1]. Lee JY, et al. Furthering pharmacological and physiological assessment of the glutamatergic receptors at the Drosophila neuromuscular junction. Comp Biochem Physiol C Toxicol Pharmacol. 2009 Nov;150(4):546-57.
Average Rating: 5 (Based on Reviews and 38 reference(s) in Google Scholar.)
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