TRPV2-selective blocker 1 |
| Katalog-Nr.GC71419 |
TRPV2-selective blocker 1 (Verbindung IV2-1) ist ein selektiver TRPV2-Kanalblocker mit einem IC50 von 6,3 μM.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2242724-49-6
Sample solution is provided at 25 µL, 10mM.
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TRPV2-selective blocker 1 (compound IV2-1) is a selective TRPV2 channel blocker with an IC50 of 6.3 μM. TRPV2-selective blocker 1 does not affect TRPV1, TRPV3 or TRPV4 channels. TRPV2-selective blocker 1 also inhibits TRPV2-mediated Ca2+ influx in macrophages, and inhibits macrophage phagocytosis.
References:
[1]. Rick Raudszus, et al. Pharmacological inhibition of TRPV2 attenuates phagocytosis and lipopolysaccharide-induced migration of primary macrophages. Br J Pharmacol. 2023 Nov;180(21):2736-2749.
Review for TRPV2-selective blocker 1
Average Rating: 5 (Based on Reviews and 30 reference(s) in Google Scholar.)
Review for TRPV2-selective blocker 1
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