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BMS-984923

Catalog No.GC68784

BMS-984923 est un régulateur allostérique efficace du silençage de mGluR5, avec une bonne affinité (Ki = 0,6 nM), une bonne biodisponibilité orale et une perméabilité à la barrière hémato-encéphalique. BMS-984923 inhibe efficacement l'interaction PrPC-mGluR5 sans affecter le signal physiologique de l'acide glutamique, tout en inhibant le signal pathologique Aβo.

Products are for research use only. Not for human use. We do not sell to patients.

BMS-984923 Chemical Structure

Cas No.: 1375752-78-5

Taille Prix Stock Qté
5mg
495,00 $US
En stock
10mg
810,00 $US
En stock

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Sample solution is provided at 25 µL, 10mM.

Chemical Properties Product Documents

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Average Rating: 5 ★★★★★ (Based on Reviews and 30 reference(s) in Google Scholar.)

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