Eact |
Catalog No.GC18142 |
Eact est un activateur sélectif et puissant de TMEM16A, active directement les canaux TRPV1 dans les nocicepteurs sensoriels et produit des démangeaisons, une nociception aiguë et une hypersensibilité thermique.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 461000-66-8
Sample solution is provided at 25 µL, 10mM.
TMEM16A (ANO1) calcium-activated chloride channel (CaCC) activator (EC50 = 3 μM). Also transient receptor potential vanilloid 1 (TRPV1) channel activator (EC50 = 11.6 μM). Ca2+-independent. Displays no effect on CFTR Cl- or ENaC Na+ conductance. Stimulates submucosal gland secretion in human bronchi.
Average Rating: 5
(Based on Reviews and 28 reference(s) in Google Scholar.)GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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