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Sigma-1 receptor antagonist 2

Catalog No.GC38039

L'antagoniste 2 des récepteurs Sigma-1 est un antagoniste puissant et sélectif des récepteurs sigma 1 (σ1 R) avec Kis de 3,88 et 1288 nM pour les récepteurs σ1 et σ2, respectivement .

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Sigma-1 receptor antagonist 2 Chemical Structure

Cas No.: 1639220-15-7

Taille Prix Stock Qté
10mM (in 1mL DMSO)
297,00 $US
En stock
1mg
202,00 $US
En stock
5mg
270,00 $US
En stock
10mg
450,00 $US
En stock

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents Related Products

Sigma-1 receptor antagonist 2 is a potent and selective sigma 1 receptor (σ1 R) antagonist with Kis of 3.88 and 1288 nM for σ1 and σ2 receptor, respectively[1].

[1]. Lan Y, et al. Synthesis and biological evaluation of novel sigma-1 receptor antagonists based on pyrimidine scaffold as agents for treating neuropathic pain. J Med Chem. 2014 Dec 26;57(24):10404-23.

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