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Glutaminase C Inhibitor 11

Catalog No.GC91427

Le inhibiteur de la glutaminase C 11 est un inhibiteur de la glutaminase C (GAC).

Products are for research use only. Not for human use. We do not sell to patients.

Glutaminase C Inhibitor 11 Chemical Structure

Taille Prix Stock Qté
1mg
111,00 $US
En stock
5mg
525,00 $US
En stock
10mg
995,00 $US
En stock

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents
Glutaminase C inhibitor 11 is an inhibitor of glutaminase C (GAC).1 It inhibits GAC enzyme activity (EC50 = 10.64 nM) and reduces the viability of A549 non-small cell lung cancer (NSCLC) cells (IC50 = 4.025 nM). Glutaminase C inhibitor 11 (0.1 and 1 µM) reduces colony formation by, and intracellular glutamate levels in, A549 cells. In vivo, glutaminase C inhibitor 11 (100 mg/kg) reduces tumor growth in an A549 mouse xenograft model.

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Average Rating: 5 ★★★★★ (Based on Reviews and 30 reference(s) in Google Scholar.)

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