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IEM 1754 dihydrobroMide

Catalog No.GC12198

IEM 1754 dihydrobroMide, un dérivé dicationique de l'adamantane, est un puissant bloqueur des canaux ouverts des récepteurs ionotropes natifs du glutamate, y compris les récepteurs sensibles au quisqualate dans les muscles des insectes, le NMDAR dans les neurones corticaux de rat en culture et l'AMPAR dans les cellules hippocampiques fraÎchement isolées.

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IEM 1754 dihydrobroMide Chemical Structure

Cas No.: 162831-31-4

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents Related Products

IEM 1754 dihydrobroMide is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.

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Average Rating: 5 ★★★★★ (Based on Reviews and 11 reference(s) in Google Scholar.)

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