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MRS 1754

Catalog No.GC13807

MRS 1754 est un radioligand antagoniste sélectif du récepteur A2B de l'adénosine avec une très faible affinité pour les récepteurs A1 et A3 des humains et des rats .

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MRS 1754 Chemical Structure

Cas No.: 264622-58-4

Taille Prix Stock Qté
10mM (in 1mL DMSO)
178,00 $US
En stock
5mg
162,00 $US
En stock
10mg
234,00 $US
En stock
25mg
504,00 $US
En stock

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Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents Related Products

MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats[1].

The most potent displacer of [3H]MRS 1754 binding is MRS 1754. The Ki value for displacement of [3H]MRS 1754 binding to human A2B receptors expressed in HEK-293 cell membranes is 1.45±0.21 nM[1].

References:
[1]. Ji X, et al. [3H]MRS 1754, a selective antagonist radioligand for A(2B) adenosine receptors. Biochem Pharmacol. 2001 Mar 15;61(6):657-63.

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