SYM 2081 |
| Catalog No.GC16101 |
SYM 2081 est un ligand de haute affinité et un puissant agoniste sélectif des récepteurs kaÏnate, inhibe la liaison [3H]-kaÏnate avec une IC50 de 35 nM, une sélectivité de près de 3000 et 200 fois pour les récepteurs kaÏnate par rapport aux récepteurs AMPA et NMDA respectivement [1 ].
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 31137-74-3
Sample solution is provided at 25 µL, 10mM.
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SYM 2081 is a high-affinity ligand and potent, selective agonist of kainate receptors, inhibits [3H]-kainate binding with an IC50 of 35 nM, almost 3000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively[1].
References:
[1]. Lee JY, et al. Furthering pharmacological and physiological assessment of the glutamatergic receptors at the Drosophila neuromuscular junction. Comp Biochem Physiol C Toxicol Pharmacol. 2009 Nov;150(4):546-57.
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