TbPTR1 inhibitor 2 |
| Catalog No.GC72510 |
TbPTR1 inhibitor 2 (composé 3a) est un inhibiteur de l’enzyme PTR1, avec des ci50 de 34,2 et 32,9 μM pour TbPTR1 et LmPTR1.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 17557-67-4
Sample solution is provided at 25 µL, 10mM.
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TbPTR1 inhibitor 2 (Compound 3a) is a PTR1 enzyme inhibitor, with IC50s of 34.2 and 32.9 μM for TbPTR1 and LmPTR1. TbPTR1 inhibitor 2 has anti-parasitic activity against T. brucei (IC50: 34.2 μM).
References:
[1]. Linciano P, et al. Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections. J Med Chem. 2019 Apr 25;62(8):3989-4012.
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