TRPV2-selective blocker 1 |
| Catalog No.GC71419 |
TRPV2-selective blocker 1 (composé iv2 - 1) est un bloqueur sélectif du canal trpv2 avec une CI50 de 6,3 µm.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2242724-49-6
Sample solution is provided at 25 µL, 10mM.
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TRPV2-selective blocker 1 (compound IV2-1) is a selective TRPV2 channel blocker with an IC50 of 6.3 μM. TRPV2-selective blocker 1 does not affect TRPV1, TRPV3 or TRPV4 channels. TRPV2-selective blocker 1 also inhibits TRPV2-mediated Ca2+ influx in macrophages, and inhibits macrophage phagocytosis.
References:
[1]. Rick Raudszus, et al. Pharmacological inhibition of TRPV2 attenuates phagocytosis and lipopolysaccharide-induced migration of primary macrophages. Br J Pharmacol. 2023 Nov;180(21):2736-2749.
Review for TRPV2-selective blocker 1
Average Rating: 5 (Based on Reviews and 30 reference(s) in Google Scholar.)
Review for TRPV2-selective blocker 1
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