iBRD4-BD1 diTFA |
Catalog No.GC71159 |
iBRD4-BD1 diTFA is selective BRD4 bromodomain inhibitor. iBRD4-BD1 diTFA has inhibition activity for BRD4 bromodomain with an IC50 value of 12 nM.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2839318-20-4
Sample solution is provided at 25 µL, 10mM.
iBRD4-BD1 diTFA has affinity and selectivity for the BET-family BRD4-BD1 with an IC50 value of 12 nM[1].
iBRD4-BD1 diTFA has affinity and selectivity for the BET-family BRD4-BD2, BRD3-BD1, BRD3-BD2, BRD2-BD1 and BRD2-BD2 with IC50 values of 16 μM, 1.0 μM , 75 μM , 280 nM and 7.1 μM, respectively[1].
iBRD4-BD1 (0-50 μM; 72 h) diTFA has cytotoxicity with an EC50 value of 2.3 μM in MM.1S cells[1].
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