5-fluoro SDB-005 |
| カタログ番号GC42538 |
5-フルオロSDB-005は、中枢のCB1受容体（EC50 = 21 nM）を望ましい方向に選択的に活性化する合成カンナビノイド（CB）であるSDB-005のアナログです。周辺のCB2受容体（EC50 = 140 nM）よりも優先的に作用します。
Products are for research use only. Not for human use. We do not sell to patients.
Sample solution is provided at 25 µL, 10mM.
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5-fluoro SDB-005 is an analog of SDB-005, a synthetic cannabinoid (CB) that activates the central CB1 receptor (EC50 = 21 nM) preferentially over the peripheral CB2 receptor (EC50 = 140 nM).[1] While the properties of this compound are not known, the addition of fluorine to the terminal carbon of the alkyl chain in similar cannabimimetic compounds typically increases affinity for both CB receptors significantly.[2] This product is intended for research and forensic applications.
Reference:
[1]. Banister, S.D., Wilkinson, S.M., Longworth, M., et al. The synthesis and pharmacological evaluation of adamantane-derived indoles: Cannabimimetic drugs of abuse. ACS Chem.Neurosci. 4(7), 1081-1092 (2013).
[2]. Makriyannis, A., and Deng, H. Cannabimimetic indole derivatives. PCT/US00/28832, (2001).
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