DL-Dapoxetine (hydrochloride) |
カタログ番号GC90686 |
(R)-ダポキセチンと(S)-ダポキセチンのラセミ混合物
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Cas No.: 1071929-03-7
Sample solution is provided at 25 µL, 10mM.
DL-Dapoxetine is a racemic mixture of the serotonin (5-HT) reuptake inhibitors (R)-dapoxetine and (S)-dapoxetine.1 (S)-Dapoxetine is more potent than (R)-dapoxetine in a serotonin reuptake assay using isolated rat cerebral cortex membranes (IC50s = 10 and 35 nM, respectively).2 (S)-Dapoxetine also inhibits the reuptake of norepinephrine and dopamine in cells expressing the human transporters (IC50s = 202 and 1,720 nM, respectively).3 Formulations containing (S)-dapoxetine have been used in the treatment of premature ejaculation.
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