(D-Pen²,p-chloro-Phe⁴,D-Pen⁵)-Enkephalin |
| カタログ番号GA20144 |
DPDPEのPhe?芳香環のパラ位にクロロ置換基を導入することで、δ-選択性が親ペプチドより5倍高くなる化合物が得られました。これは、δ-受容体親和性が5倍増加したためです。(Cpa?)-DPDPEは、この理由から、δ-オピオイド受容体の特性を研究するための最適なリガンドとなる可能性があります。
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 122507-47-5
Sample solution is provided at 25 µL, 10mM.
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The introduction of a chloro substituent in para-position of the Phe aromatic ring of DPDPE led to a compound with 5 times higher δ-selectivity than the parent peptide due to a 5-fold increased δ-receptor affinity. For this reason, (Cpa)-DPDP
Average Rating: 5 (Based on Reviews and 16 reference(s) in Google Scholar.)
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