4-Abz-Gly-Pro-D-Leu-D-Ala-NHOH |
カタログ番号GA20408 |
水溶性ペプチドヒドロキサム酸FN439は、人間のマトリックスメタロプロテアーゼの広範なスペクトル阻害剤です。4-Abz-Gly-Pro-D-Leu-D-Ala-NHOHは、プロナーゼまたはヒト顆粒球エラスターゼと長時間培養しても活性を保持します。FN 439は、間質性および顆粒球コラゲナーゼ、顆粒球ゲラチナーゼおよび皮膚線維芽細胞ストロメリシンをそれぞれ1.10?? M、3.10?? Mおよび1.5.10?? MのIC50で阻害します。
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Cas No.: 124168-73-6
Sample solution is provided at 25 µL, 10mM.
The water-soluble peptidylhydroxamic acid FN439 is a broad-spectrum inhibitor of human matrix metalloproteinases. 4-Abz-Gly-Pro-D-Leu-D-Ala-NHOH retains its activity even after prolonged incubation with pronase or human granulocyte elastase. FN 439 inh
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