BIM-23627 |
カタログ番号GA20812 |
ソマトスタチン拮抗剤BIM 23627は、高親和性で人間のソマトスタチン受容体サブタイプ2(hsst2)に選択的に結合しますが、細胞内カルシウム動員を刺激することは完全に無効でした。 BIM 23627のIC??値は、5つの人間のソマトスタチン受容体サブタイプに対して次のようになります:2757 nM(hsst1)、6.4 nM(hsst2)、44 nM(hsst3)、423 nM(hsst4)および86.5 nM( hsst5)。
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Cas No.: 429619-37-4
Sample solution is provided at 25 µL, 10mM.
The somatostatin antagonist BIM 23627 selectively bound with high affinity to the human somatostatin receptor subtype 2 (hsst2), but was completely inactive in stimulating intracellular calcium mobilization. The IC50 values of BIM 23627 to the five hum
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