MRS 1754 |
カタログ番号GC13807 |
MRS 1754 は、ヒトとラットの両方の A1 および A3 受容体に対する親和性が非常に低い、A2B アデノシン受容体に対する選択的アンタゴニスト放射性リガンドです 。
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Cas No.: 264622-58-4
Sample solution is provided at 25 µL, 10mM.
MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats[1].
The most potent displacer of [3H]MRS 1754 binding is MRS 1754. The Ki value for displacement of [3H]MRS 1754 binding to human A2B receptors expressed in HEK-293 cell membranes is 1.45±0.21 nM[1].
References:
[1]. Ji X, et al. [3H]MRS 1754, a selective antagonist radioligand for A(2B) adenosine receptors. Biochem Pharmacol. 2001 Mar 15;61(6):657-63.
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