Repinotan hydrochloride (Synonyms: BAY x 3702) |
| カタログ番号GC64423 |
レピノタン塩酸塩 (BAY x 3702) は、強力で選択的な脳浸透型の経口活性 5-HT1A 受容体アゴニストであり、Ki 値は 0.19 nM (子牛の海馬)、0.25 nM (ラットおよびヒトの皮質)、および 0.59 nM (ラットの海馬 レピノタン塩酸塩は、他の関連する受容体に対して弱い親和性を持っています。
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 144980-77-8
Sample solution is provided at 25 µL, 10mM.
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Repinotan hydrochloride (BAY x 3702) is a potent, selective, brain-penetrant and orally active 5-HT1A receptor agonist, with Ki values of 0.19 nM (calf hippocampus), 0.25 nM (rat and human cortex), and 0.59 nM (rat hippocampus Repinotan hydrochloride has a weak affinity for other related receptors. Repinotan hydrochloride has pronounced neuroprotective effects[1].
[1]. A C Berends, et al. A review of the neuroprotective properties of the 5-HT1A receptor agonist repinotan HCl (BAYx3702) in ischemic stroke. CNS Drug Rev. Winter 2005;11(4):379-402.
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