CB2R-IN-1 |
カタログ番号GC33756 |
CB2R-IN-1 は、Ki が 0.9 nM の強力なカンナビノイド CB2 受容体逆アゴニストです。
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1257555-79-5
Sample solution is provided at 25 µL, 10mM.
CB2R-IN-1 is a potent cannabinoid CB2 receptor inverse agonist with a Ki of 0.9 nM.
CB2R-IN-1 (Compound 37) is a potent cannabinoid CB2 receptor ligand (Ki=0.9 nM) with excellent selectivity over the CB1 receptor (Ki=8259.3 nM)[1].
[1]. Tong L, et al. Expansion of SAR studies on triaryl bis sulfone cannabinoid CB2 receptor ligands. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6785-9.
Average Rating: 5
(Based on Reviews and 2 reference(s) in Google Scholar.)GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.
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