RXR antagonist 1 |
| カタログ番号GC70895 |
RXR antagonist 1（化合物6 a）は、レチノイン酸X受容体（RXR）調整剤である。
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 3010910-40-1
Sample solution is provided at 25 µL, 10mM.
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RXR antagonist 1 (compound 6a) is a retinoid X receptor (RXR) modulator. RXR antagonist 1 shows potent RXR-antagonistic activity, with a pA2 of 8.06. RXR antagonist 1 can be used for type 2 diabetes research.
RXR antagonist 1 (compound 6a) shows potent RXR-antagonistic activities at 1 μM[1].
RXR antagonist 1 shows competitive binding to the LBP in hRXRα-LBD, with Ki of 0.384 ± 0.072, Kd of 0.277 ± 0.038, and Ki/Kd of 1.39[1].
The cell permeability of RXR antagonist 1 shows no correlation with RXR-antagonistic activity[1].
Review for RXR antagonist 1
Average Rating: 5 (Based on Reviews and 30 reference(s) in Google Scholar.)
Review for RXR antagonist 1
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