CB1/2 agonist 3 |
Catalog No.GC71112 |
CB1/2 agonist 3 (화합물 52) 는 강력한 비선택적 대마초 배합체로 CB1/CB2 (대마초 수용체) 경쟁 흥분제입니다.
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Cas No.: 2772655-86-2
Sample solution is provided at 25 µL, 10mM.
CB1/2 agonist 3 (compound 52) can partially induce [35S]GTPγS binding to hCB1-CHO cell membranes with an EC50 value of 30.99 nM, and slightly inhibit [35S]GTPγS binding to hCB2-CHO cell membranes with a mean EC50 value of 1.28 nM[1].
CB1/2 agonist 3 (compound 52) ((1 μM, 1 h) has antagonistic effect on CB1/CB2 agonist CP-55940 with a Kb value of 78.17 nM[1].
References:
[1]. Antonella Brizzi, et al. Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity. Bioorg Med Chem. 2020 Jun 1;28(11):115513.
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