>>Signaling Pathways>> Chromatin/Epigenetics>> Epigenetic Reader Domain>>iBRD4-BD1 diTFA

iBRD4-BD1 diTFA

Catalog No.GC71159

iBRD4-BD1 diTFA 는 선택적 BRD4 브롬 구조역 억제제입니다. iBRD4-BD1 diTFABRD4 브롬 구조 도메인에 대한 억제 활성, IC50 값은 12nM입니다.

Products are for research use only. Not for human use. We do not sell to patients.

iBRD4-BD1 diTFA Chemical Structure

Cas No.: 2839318-20-4

Size 가격 재고 수량
1 mg
US$297.00
재고 있음
5 mg
US$743.00
재고 있음

Tel:(909) 407-4943 Email: sales@glpbio.com

고객 리뷰

Based on customer reviews.

  • GlpBio Citations

    GlpBio Citations
  • Bioactive Compounds Premium Provider

    Bioactive Compounds Premium Provider

Sample solution is provided at 25 µL, 10mM.

Description Chemical Properties Product Documents
iBRD4-BD1 diTFA is selective BRD4 bromodomain inhibitor. iBRD4-BD1 diTFA has inhibition activity for BRD4 bromodomain with an IC50 value of 12 nM. iBRD4-BD1 diTFA can be used for the research of inflammation and oncology.

iBRD4-BD1 diTFA has affinity and selectivity for the BET-family BRD4-BD1 with an IC50 value of 12 nM[1].
iBRD4-BD1 diTFA has affinity and selectivity for the BET-family BRD4-BD2, BRD3-BD1, BRD3-BD2, BRD2-BD1 and BRD2-BD2 with IC50 values of 16 μM, 1.0 μM , 75 μM , 280 nM and 7.1 μM, respectively[1].
iBRD4-BD1 (0-50 μM; 72 h) diTFA has cytotoxicity with an EC50 value of 2.3 μM in MM.1S cells[1].

리뷰

Review for iBRD4-BD1 diTFA

Average Rating: 5 ★★★★★ (Based on Reviews and 30 reference(s) in Google Scholar.)

5 Star
100%
4 Star
0%
3 Star
0%
2 Star
0%
1 Star
0%
Review for iBRD4-BD1 diTFA

GLPBIO products are for RESEARCH USE ONLY. Please make sure your review or question is research based.

Required fields are marked with *

You may receive emails regarding this submission. Any emails will include the ability to opt-out of future communications.