iBRD4-BD1 diTFA |
Catalog No.GC71159 |
iBRD4-BD1 diTFA 는 선택적 BRD4 브롬 구조역 억제제입니다. iBRD4-BD1 diTFABRD4 브롬 구조 도메인에 대한 억제 활성, IC50 값은 12nM입니다.
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Cas No.: 2839318-20-4
Sample solution is provided at 25 µL, 10mM.
iBRD4-BD1 diTFA has affinity and selectivity for the BET-family BRD4-BD1 with an IC50 value of 12 nM[1].
iBRD4-BD1 diTFA has affinity and selectivity for the BET-family BRD4-BD2, BRD3-BD1, BRD3-BD2, BRD2-BD1 and BRD2-BD2 with IC50 values of 16 μM, 1.0 μM , 75 μM , 280 nM and 7.1 μM, respectively[1].
iBRD4-BD1 (0-50 μM; 72 h) diTFA has cytotoxicity with an EC50 value of 2.3 μM in MM.1S cells[1].
Average Rating: 5
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