PROTAC ERRα ligand 2 |
| Catalog No.GC38383 |
PROTAC ERRα 리간드 2는 5.67 nM의 IC50을 갖는 에스트로겐 관련 수용체 α(ERRα) 역 작용제입니다. PROTAC ERRα 리간드 2(IC50\u003d5.67nM)는 XCT790(IC50\u003d61.3nM)보다 ~11배 향상된 효능을 나타냅니다.
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Cas No.: 2306388-57-6
Sample solution is provided at 25 µL, 10mM.
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PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist with an IC50 of 5.67 nM. PROTAC ERRα ligand 2 (IC50=5.67 nM) displays a ~11-fold improved potency than XCT790 (IC50=61.3 nM)[1].
[1]. Peng L, et al. Identification of New Small-Molecule Inducers of Estrogen-related Receptor α (ERRα) Degradation. ACS Med Chem Lett. 2019 Apr 12;10(5):767-772.
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