Elacestrant (S enantiomer) (Synonyms: RAD1901 S enantiomer) |
| Catalog No.GC62379 |
El enantiÓmero S de Elacestrant (enantiÓmero RAD1901 S) es un enantiÓmero de baja actividad de Elacestrant. Elacestrant (RAD1901) es un degradador del receptor de estrÓgeno (ERR) selectivo y disponible por vÍa oral con valores IC50 de 48 y 870 nM para ERα y ERβ, respectivamente.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2309762-29-4
Sample solution is provided at 25 µL, 10mM.
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Elacestrant S enantiomer (RAD1901 S enantiomer) is an low activity enantiomer of elacestrant. Elacestrant (RAD1901) is a selective and orally available estrogen receptor (ERR) degrader with IC50 values of 48 and 870 nM for ERα and ERβ, respectively[1].
[1]. Garner F, et al. RAD1901: a novel, orally bioavailable selective estrogen receptor degrader that demonstrates antitumor activity in breast cancer xenograft models. Anticancer Drugs. 2015 Oct;26(9):948-56.
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