GX 201 |
| Catalog No.GC50707 |
GX 201 es un inhibidor selectivo de NaV1.7, con una IC50 de \u003c3,2 nM para hNaV1.7.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 1788071-27-1
Sample solution is provided at 25 µL, 10mM.
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Potent and selective Nav1.7 blocker (IC50 = 3.2 nM). Exhibits 10x selectivity for Nav1.7 over Nav1.1, Nav1.2, and Nav1.6 channels. Displays prolonged residency time on the Nav1.7 channel. Chronic dosing increases compound potency ~10-fold and provides efficacy that persists after the compound has cleared from plasma. Suppresses neuropathic pain in a mouse diabetic neuropathy model. Analgesic.
Average Rating: 5 (Based on Reviews and 7 reference(s) in Google Scholar.)
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