LPA2 antagonist 2 |
| Catalog No.GC38923 |
El antagonista 2 de LPA2 (H2L 5226501) es un antagonista selectivo de LPA2 con una CI50 de 28,3 nM y una Ki de 21,1 nM. El antagonista 2 de LPA2 es >480 veces mÁs selectivo que LPA3 (IC50 de 13,85 μM).
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Cas No.: 36840-10-5
Sample solution is provided at 25 µL, 10mM.
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LPA2 antagonist 2 (H2L 5226501) is a selective LPA2 antagonist with an IC50 of 28.3 nM, which is ＞480-fold more selective than LPA3 (IC50 of 13.85 μM)[1].
[1]. Fells JI, et al. Identification of non-lipid LPA3 antagonists by virtual screening. Bioorg Med Chem. 2008 Jun 1;16(11):6207-17.
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