OXFBD04 |
| Catalog No.GC39417 |
OXFBD04 es un inhibidor de BRD4 potente y selectivo con una IC50 de 166 nM. OXFBD04 es un potente ligando de bromodominio BET con una modesta afinidad adicional por el bromodominio CREBBP. OXFBD04 tiene actividad anticancerÍgena.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 2231747-03-6
Sample solution is provided at 25 µL, 10mM.
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OXFBD04 is a potent and selective BRD4 inhibitor with an IC50 of 166?nM. OXFBD04 is a potent BET bromodomain ligand with additional modest affinity for the CREBBP bromodomain. OXFBD04 has anti-cancer activity[1].
[1]. Jennings LE, et al. BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability. Bioorg Med Chem. 2018 Jul 15;26(11):2937-2957.
Average Rating: 5 (Based on Reviews and 24 reference(s) in Google Scholar.)
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