LAS101057 |
| Catalog No.GC33871 |
LAS101057 es un antagonista del receptor A2B potente, selectivo y eficaz por vÍa oral.
Products are for research use only. Not for human use. We do not sell to patients.
Cas No.: 925676-48-8
Sample solution is provided at 25 µL, 10mM.
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LAS101057 is a potent, selective, and orally efficacious A2B receptor antagonist.
At 3 mg/kg, LAS101057 is active in preventing methacholine-induced AHR, and at 10 mg/kg it inhibits AHR to methacholine to a level virtually equal to that seen with dexamethasone at 1 mg/kg[1].
[1]. Paul Eastwood, et al. Discovery of LAS101057: A Potent, Selective, and Orally Efficacious A2B Adenosine Receptor Antagonist. ACS Med Chem Lett. 2011 Mar 10; 2(3): 213-218.
Average Rating: 5 (Based on Reviews and 39 reference(s) in Google Scholar.)
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